Fascaplysin-inspired diindolyls as selective inhibitors of CDK4/cyclin D1

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Aubry, C., Wilson, A.J., Emmerson D., Murphy, E., Chan, Y.Y., Dickens, M.P., García, M.D., Jenkins, P.R., Mahale, S., Chaudhuri, B. (2009) Fascaplysin-inspired diindolyls as selective inhibitors of CDK4/cyclin D1. Bioorganic & Medicinal Chemistry, 17 (16) pp. 6073-84.

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Research Institute