Browsing School of Allied Health Sciences by Subject "partial agonism"
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Predicting in vivo cardiovascular properties of blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses (Article)Beta -Adrenoceptor antagonists differ in their degree of partial agonism. In vitro assays have provided information on ligand affinity, selectivity, and intrinsic efficacy. However, the extent to which these properties are ...